Androgen Receptor
AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.
- A2150 AndarineTarget: Androgen ReceptorsSummary: Androgen receptor agonist
- A8364 ARN-5092 CitationTarget: Androgen ReceptorSummary: Androgen receptor inhibitor
- A8452 ODM-201Target: Androgen ReceptorsSummary: new-generation androgen receptor inhibitor
- B1505 EpiandrosteroneTarget: Voltage-gated Calcium Channels (CaV)Summary: steroid hormone with weak androgenic activity
- B1506 Estradiol valerateTarget: Estrogen and Related ReceptorsSummary: Estrogen receptor agonist
- B7468 CITCO1 CitationTarget: constitutive androstane receptor (CAR)Summary: A selective constitutive androstane receptor (CAR) agonist
- A3003 MDV3100 (Enzalutamide)12 CitationTarget: Androgen ReceptorsSummary: Androgen receptor antagonist
- A4326 TAK-700 (Orteronel)2 CitationTarget: human lyaseSummary: Human 17,20-lyase inhibitor
- A3190 ASC-J9Summary: AR degradation enhancer,antiumor agent