Signaling Pathways
- A5065 Bicalutamide1 CitationTarget: Androgen ReceptorsSummary: Androgen receptor antagonist
- A8623 TOK-001Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17 inhibitor and androgen receptor (AR) antagonist
- B3238 XCT790Target: Estrogen and Related ReceptorsSummary: ERRα agonist
- B1515 Raloxifene HClTarget: Estrogen and Related ReceptorsSummary: Estrogen receptor (ER)
- B5421 (Z)-4-HydroxytamoxifenTarget: Estrogen and Related ReceptorsSummary: ER modulator, potent and selective
- B5455 G-14 CitationTarget: GPR30Summary: GPR30 agonist, potent and selective
- B5469 G-153 CitationTarget: GPR30Summary: GPER receptor antagonist
- B1518 Erteberel (LY500307)Target: Estrogen and Related ReceptorsSummary: ERβ agonist, potent and selective
- B1510 Medroxyprogesterone acetateTarget: Progesterone ReceptorsSummary: Steroidal progestin
- B6429 Naltrindole hydrochlorideSummary: δ opioid antagonist