VEGFR
VEGFR are receptors for vascular endothelial growth factor and belong to receptor tyrosine kinases.
- A8550 Telatinib (BAY 57-9352)Target: VEGFR|PDGFR|c-KitSummary: VEGFR-2/-3,PDGFR-β and c-Kit inhibitor
- A8555 Vandetanib (ZD6474)Target: VEGFR|EGFRSummary: VEGFR2/EGFR antagonist
- B1305 SKLB1002Summary: VEGFR2 inhibitor,potent and ATP-competitve
- B2173 CP-673451Target: PDGFRSummary: PDGFRα/β inhibitor,potent and selective
- B2303 Apatinib1 CitationSummary: VEGFR2 inhibitor, orally bioavailable, selective
- B6199 BFH772Summary: VEGFR2 inhibitor
- B7800 BAW2881 (NVP-BAW2881)Summary: VEGFR inhibitor
- C3342 MAZ51Target: VEGFRSummary: VEGFR3 antagonist
- C3415 Tivozanib (hydrate)Summary: VEGFR inhibitor, orally available
- C3730 AAL-993Summary: VEGF receptors inhibitor