HER2
HER2 is a member of the epidermal growth factor. It initiates the EGF downstream cascade by forming a heterodimer with other ligand-bound EGF receptor. It is associated with breast and ovarian cancers.
- A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: Multitargeted HDAC inhibitor
- A3145 Afatinib dimaleateTarget: EGFR|HER2Summary: EGFR inhibitor
- A3252 BMS-599626 HydrochlorideSummary: EGFR/HER2 inhibitor,potent and selective
- A3276 Canertinib dihydrochlorideSummary: Pan-ErbB inhibitor, potent and selective