Signaling Pathways
- A8706 BLU9931Target: FGFRSummary: FGFR4 inhibitor,potent and irreversible
- A3009 Sorafenib2 CitationTarget: Raf|VEGFRSummary: Raf kinases and tyrosine kinases inhibitor
- A3014 BGJ3981 CitationTarget: FGFRSummary: FGFR inhibitor ,potent and selective
- A3020 (R)-Crizotinib2 CitationTarget: c-METSummary: C-MET/ALK inhibitor,potent and ATP-competitve
- A3022 Pazopanib (GW-786034)Target: CSF-1R|VEGFR|PDGFR|c-Kit|FGFRSummary: VEGFR/PDGFR/FGFR inhibitor
- A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: Multitargeted HDAC inhibitor
- A4139 AG-4903 CitationTarget: EGFR|JAKSummary: JAK2/EGFR inhibitor
- A4116 Danusertib (PHA-739358)2 CitationTarget: Aurora KinasesSummary: Pan-aurora kinase inhibitor
- A3145 Afatinib dimaleateTarget: EGFR|HER2Summary: EGFR inhibitor
- A3194 AST 4871 CitationTarget: RETSummary: RET kinase inhibitor