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5-HT Receptor

5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.

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  1. Cat.No. Product Name Information
  2. B2237 Eletriptan HBr selective 5-HT1B and 5-HT1D receptor agonist
  3. B2236 Desvenlafaxine serotonin (5-HT) and norepinephrine (NE) reuptake inhibitor
  4. B2246 Desvenlafaxine Succinate serotonin (5-HT) transporter and norepinephrine (NE) transporter reuptake inhibitor
  5. B2250 LY310762 5-HT1D receptor antagonist
  6. B2253 Prucalopride 5-HT4A and 5-HT4B receptor agonist
  7. B2255 SB271046 5-HT6 receptor antagonist, orally active
  8. B2259 VUF 10166 5-HT3 receptor antagonist
  9. B2260 WAY-100635 Maleate 5-HT1A receptor agonist
  10. B2233 Azasetron HCl 5-HT3 receptor antagonist
  11. B2243 Almotriptan Malate 5-HT1B/1D-receptor agonist
  12. B2241 Ondansetron serotonin 5-HT3 receptor antagonist
  13. B2230 Trazodone HCl 5-HT receptor antagonist
  14. B2234 Clomipramine HCl SERT/NET dopamine transporter (DAT) blocker
  15. B2263 BMY 7378 5-HT1A partial agonist and α1D adrenoceptor antagonist
  16. B2231 Amitriptyline HCl Serotonin /norepinephrine receptor/5-HT4/5-HT2 inhibitor
  17. B2229 Palonosetron HCl 5-HT receptor antagonist
  18. B1754 Fenspiride HCl α adrenergic and H1 histamine receptor antagonist
  19. B1204 Ondansetron hydrochloride dihydrate 5-HT3 receptor antagonist
  20. B1002 Tropisetron Hydrochloride 5-HT3 receptor antagonist
  21. B1477 Lurasidone HCl Dopamine D2/5-HT2A/5-HT7/5-HT1A inhibitor
  22. B2258 Tropisetron 5-HT3 receptor antagonist
  23. B1205 Fluvoxamine Selective serotonin reuptake inhibitor
  24. B1206 Pizotifen Highly selective 5-HT receptor blocking agent
  25. B2007 Pizotifen Malate 5-HT receptor antagonist
  26. B1059 Mosapride Selective 5HT4 agonist
  27. B2251 Naratriptan selective 5-HT1 receptor subtype agonist
  28. B2261 Zolmitriptan Potent 5-HT1B/1D/1F agonist
  29. B2242 Urapidil HCl α1-adrenoceptor antagonist and 5-HT1A receptor agonist
  30. B2264 Dapoxetine HCl Selective serotonin reuptake inhibitor
  31. B6659 (S)-WAY 100135 dihydrochloride 5-HT1A receptor antagonist,potent and selective
  32. B6736 Citalopram hydrobromide 5-HT uptake inhibitor
  33. B6799 Indatraline hydrochloride Inhibits transporters for 5-HT (SERT), dopamine (DAT) and noradrenalin (NET)
  34. B6851 Zimelidine dihydrochloride 5-HT re-uptake inhibitor
  35. B6852 S 14506 hydrochloride 5-HT1A receptor full agonist
  36. B6883 Ipsapirone 5-HT1A receptor agonist
  37. B6952 Paroxetine maleate 5-HT uptake inhibitor
  38. B6954 (±)-McN 5652 5-HT uptake inhibitor
  39. B7097 Lofepramine Serotonin and noradrenalin re-uptake inhibitor (SNRI)
  40. B5292 BTS 54-505 hydrochloride Potent SNRI,sibutramine metabolite
  41. B5406 NAD 299 hydrochloride Selective, high affinity 5-HT1A receptor antagonist
  42. B5538 WY 45233 succinate serotonin and noradrenalin reuptake inhibitor
  43. B6588 (R)-(+)-8-Hydroxy-DPAT hydrobromide 5-HT1A serotonin receptor agonist
  44. B6538 Cyanopindolol hemifumarate 5-HT1A/1B antagonist and β-adrenoceptor antagonist
  45. B2248 Ketanserin specific 5-HT2A serotonin receptor antagonist
  46. B6292 MDL 73005EF hydrochloride 5-HT1A receptor antagonist
  47. B6293 MDL 72832 hydrochloride ligand for 5-HT1A receptor, potent and selective
  48. B6337 8-Hydroxy-DPAT hydrobromide 5-HT1A agonist
  49. B6349 NAN-190 hydrobromide 5-HT1A antagonist
  50. B6351 BP 554 maleate Selective 5-HT1A agonist
  51. B6388 CGS 12066B dimaleate 5-HT1B full agonist
  52. B6410 Anpirtoline hydrochloride 5-HT1B receptor agonist
  53. B6457 8-Hydroxy-PIPAT oxalate 5-HT1A receptor agonist
  54. B6496 5-Nonyloxytryptamine oxalate 5-HT1B agonist
  55. B6511 MM 77 dihydrochloride 5-HT1A receptor antagonist
  56. B6537 Isamoltane hemifumarate 5-HT1B antagonist
  57. B5366 (±)-MDMA hydrochloride inhibitor of 5-HT and dopamine uptake
  58. B1203 Iloperidone hydrochloride D(2)/5-HT(2) receptor antagonistis
  59. A3144 Adoprazine 5-HT1A receptor agonist and full D2/3 receptor antagonist
  60. A3796 SB-269970 5-HT7 receptor antagonist
  61. A3811 SEA0400 Specific inhibitor of Na+/Ca2+ exchange
  62. A3873 Tianeptine 5-HT facilitator
  63. A3918 Vilazodone Combined SSRI and 5-HT1A receptor partial agonist
  64. A3919 Vilazodone Hydrochloride Combined SSRI and 5-HT1A receptor partial agonist
  65. A3926 Vortioxetine 5-HT receptors antagonist
  66. A3933 WAY-100635 5-HT1A receptor antagonist,potent and selective
  67. A3934 WAY-100635 maleate salt 5-hydroxytryptamine 1A antagonist
  68. A3952 Ziprasidone 5-HT (serotonin)/dopamine receptor antagonist
  69. A3953 Ziprasidone hydrochloride monohydrate 5-HT (serotonin)/dopamine receptor antagonist
  70. A1295 Granisetron HCl 5-HT3 receptor antagonist
  71. A1334 Mosapride Citrate 5-HT receptor agonist
  72. A3778 RS 127445 5-HT2B receptor antagonist,high affinity
  73. A3697 Palonosetron 5-HT3 antagonist
  74. A3157 Alosetron 5-HT3 receptor antagonist
  75. A3158 Alosetron (Z)-2-butenedioate 5-HT3 receptor antagonist
  76. A3159 Alosetron Hydrochloride 5-HT3 receptor antagonist,potent and highly selective
  77. A3160 Alosetron Hydrochloride(1:X) 5-HT3 receptor antagonist
  78. A3192 Asenapine hydrochloride Atypical antipsychotic
  79. A3239 B-HT 920 D2 receptor agonist
  80. A3241 Bilobalide Neuroprotective agent
  81. A3317 Clozapine N-oxide (CNO) Metabolite of clozapine, used in chemogenetics.
  82. A3330 CP-809101 5-HT2C receptor agonist
  83. A3331 CP-809101 hydrochloride 5-HT2C receptor agonist, potent and selective
  84. A3443 Granisetron Serotonin 5-HT3 receptor antagonist
  85. A3569 LY 344864 5-HT1F receptor agonist,potent and selective
  86. A5010 Asenapine Inhibits adrenergic receptor/5-HT receptor
  87. B1001 Loxapine 5-HT receptor antagonist
  88. B2265 BRL-15572 5-HT1D receptor antagonist
  89. B2245 BRL-54443 5-HT1E/1F receptor agonist,potent and selective
  90. B1198 Cisapride 5-HT4 receptor agonist
  91. B2256 SB742457 5-HT6 receptor antagonist,highly selective and high affinity
  92. B2240 Olanzapine Antagonist of 5-HT2A and dopamine D2 receptors
  93. B1199 Tandospirone Anxiolytic and antidepressant reagent
  94. B1058 Lasmiditan 5-HT1F receptor agonist
  95. B2254 SB269970 HCl 5-HT7 receptor antagonist,potent and selective
  96. B1200 PRX-08066 5-HT2BR antagonist
  97. B2262 Agomelatine MT1/MT2 / 5-HT2C agonist
  98. B1201 Agomelatine hydrochloride Norepinephrine-dopamine disinhibitor (NDDI)
  99. B1202 Agomelatine L(+)-Tartaric acid Norepinephrine-dopamine disinhibitor (NDDI)
  100. B1197 Risperidone mesylate 5-HT2 receptor blocker
  101. B1196 Risperidone hydrochloride 5-HT2 receptor blocker
  102. A2436 Fluoxetine HCl Serotonin reuptake inhibitor,selective
  103. A2553 Fluvoxamine maleate Serotonin reuptake inhibitor,selective,antidepressant
  104. A5355 Venlafaxine Dual serotonin/noradrenalin re-uptake inhibitor
  105. A5322 Tianeptine sodium 5-HT uptake facilitator,selective,antidepressant
  106. A5294 Sumatriptan Succinate 5-HT1 receptor agonist
  107. A5350 Ziprasidone HCl Serotonin and dopamine receptor antagonist
  108. A5399 Iloperidone Dopamine (D2) and serotonin (5HT2) receptor antagonist
  109. A2547 Vortioxetine (Lu AA21004) HBr 5-HT receptor modulator, antidepressant and anxiolytic
  110. A2098 PRX-08066 Maleic acid 5-HT2B receptor antagonist,potent and selective
  111. A8514 Risperidone SR-2A inhibitor
  112. A8516 Rizatriptan Benzoate 5-HT Receptor agonist
  113. A8384 Blonanserin Atypical antipsychotic
  114. A8421 Duloxetine HCl 5-HT receptor inhibitor
  115. C4117 Imipramine (hydrochloride) serotonin and norepinephrine transporters inhibitor
  116. C4077 Nortriptyline (hydrochloride) norepinephrine and serotonin transporters blocker
  117. B7848 RS 127445 HCl 5-HT2B receptor antagonist,high affinity
  118. C5214 6-fluoro-DL-Tryptophan serotonin (5-HT) synthesis inhibitor
  119. C5271 AL 34662 potent 5-HT2 receptor agonist
  120. B4981 Sumatriptan 5-HT1 receptor agonist
  121. A5166 Ondansetron HCl 5-HT3 receptor antagonist
  122. A3793 SB 271046 hydrochloride Selective 5-HT6 antagonist
  123. A3777 Rotigotine hydrochloride Agonist of dopamine D2/D3 receptor
  124. A3776 Rotigotine Agonist of dopamine D2/D3 receptor
  125. A3748 rac-Rotigotine Hydrochloride Agonist of dopamine D2/D3 receptor
  126. A3561 Lu AE58054 Hydrochloride 5-HT(6)R antagonist
  127. A3560 Lu AE58054 5-HT(6)R antagonist
  128. C5582 3,4-dihydro Naratriptan selective serotonin 5-HT1B agonist