5-HT Receptor

Cat.No. Product Name Information

B2237 Eletriptan HBr selective 5-HT1B and 5-HT1D receptor agonist

B2236 Desvenlafaxine serotonin (5-HT) and norepinephrine (NE) reuptake inhibitor

B2246 Desvenlafaxine Succinate serotonin (5-HT) transporter and norepinephrine (NE) transporter reuptake inhibitor

B2250 LY310762 5-HT1D receptor antagonist

B2253 Prucalopride 5-HT4A and 5-HT4B receptor agonist

B2255 SB271046 5-HT6 receptor antagonist, orally active

B2259 VUF 10166 5-HT3 receptor antagonist

B2260 WAY-100635 Maleate 5-HT1A receptor agonist

B2233 Azasetron HCl 5-HT3 receptor antagonist

B2243 Almotriptan Malate 5-HT1B/1D-receptor agonist

B2241 Ondansetron serotonin 5-HT3 receptor antagonist

B2230 Trazodone HCl 5-HT receptor antagonist

B2234 Clomipramine HCl SERT/NET dopamine transporter (DAT) blocker

B2263 BMY 7378 5-HT1A partial agonist and α1D adrenoceptor antagonist

B2231 Amitriptyline HCl Serotonin /norepinephrine receptor/5-HT4/5-HT2 inhibitor

B2229 Palonosetron HCl 5-HT receptor antagonist

B1754 Fenspiride HCl α adrenergic and H1 histamine receptor antagonist

B1204 Ondansetron hydrochloride dihydrate 5-HT3 receptor antagonist

B1002 Tropisetron Hydrochloride 5-HT3 receptor antagonist

B1477 Lurasidone HCl Dopamine D2/5-HT2A/5-HT7/5-HT1A inhibitor

B2258 Tropisetron 5-HT3 receptor antagonist

B1205 Fluvoxamine Selective serotonin reuptake inhibitor

B1206 Pizotifen Highly selective 5-HT receptor blocking agent

B2007 Pizotifen Malate 5-HT receptor antagonist

B1059 Mosapride Selective 5HT4 agonist

B2251 Naratriptan selective 5-HT1 receptor subtype agonist

B2261 Zolmitriptan Potent 5-HT1B/1D/1F agonist

B2242 Urapidil HCl α1-adrenoceptor antagonist and 5-HT1A receptor agonist

B2264 Dapoxetine HCl Selective serotonin reuptake inhibitor

B6659 (S)-WAY 100135 dihydrochloride 5-HT1A receptor antagonist,potent and selective

B6736 Citalopram hydrobromide 5-HT uptake inhibitor

B6799 Indatraline hydrochloride Inhibits transporters for 5-HT (SERT), dopamine (DAT) and noradrenalin (NET)

B6851 Zimelidine dihydrochloride 5-HT re-uptake inhibitor

B6852 S 14506 hydrochloride 5-HT1A receptor full agonist

B6883 Ipsapirone 5-HT1A receptor agonist

B6952 Paroxetine maleate 5-HT uptake inhibitor

B6954 (±)-McN 5652 5-HT uptake inhibitor

B7097 Lofepramine Serotonin and noradrenalin re-uptake inhibitor (SNRI)

B5292 BTS 54-505 hydrochloride Potent SNRI,sibutramine metabolite

B5406 NAD 299 hydrochloride Selective, high affinity 5-HT1A receptor antagonist

B5538 WY 45233 succinate serotonin and noradrenalin reuptake inhibitor

B6588 (R)-(+)-8-Hydroxy-DPAT hydrobromide 5-HT1A serotonin receptor agonist

B6538 Cyanopindolol hemifumarate 5-HT1A/1B antagonist and β-adrenoceptor antagonist

B2248 Ketanserin specific 5-HT2A serotonin receptor antagonist

B6292 MDL 73005EF hydrochloride 5-HT1A receptor antagonist

B6293 MDL 72832 hydrochloride ligand for 5-HT1A receptor, potent and selective

B6337 8-Hydroxy-DPAT hydrobromide 5-HT1A agonist

B6349 NAN-190 hydrobromide 5-HT1A antagonist

B6351 BP 554 maleate Selective 5-HT1A agonist

B6388 CGS 12066B dimaleate 5-HT1B full agonist

B6410 Anpirtoline hydrochloride 5-HT1B receptor agonist

B6457 8-Hydroxy-PIPAT oxalate 5-HT1A receptor agonist

B6496 5-Nonyloxytryptamine oxalate 5-HT1B agonist

B6511 MM 77 dihydrochloride 5-HT1A receptor antagonist

B6537 Isamoltane hemifumarate 5-HT1B antagonist

B5366 (±)-MDMA hydrochloride inhibitor of 5-HT and dopamine uptake

B1203 Iloperidone hydrochloride D(2)/5-HT(2) receptor antagonistis

A3144 Adoprazine 5-HT1A receptor agonist and full D2/3 receptor antagonist

A3796 SB-269970 5-HT7 receptor antagonist

A3811 SEA0400 Specific inhibitor of Na+/Ca2+ exchange

A3873 Tianeptine 5-HT facilitator

A3918 Vilazodone Combined SSRI and 5-HT1A receptor partial agonist

A3919 Vilazodone Hydrochloride Combined SSRI and 5-HT1A receptor partial agonist

A3926 Vortioxetine 5-HT receptors antagonist

A3933 WAY-100635 5-HT1A receptor antagonist,potent and selective

A3934 WAY-100635 maleate salt 5-hydroxytryptamine 1A antagonist

A3952 Ziprasidone 5-HT (serotonin)/dopamine receptor antagonist

A3953 Ziprasidone hydrochloride monohydrate 5-HT (serotonin)/dopamine receptor antagonist

A1295 Granisetron HCl 5-HT3 receptor antagonist

A1334 Mosapride Citrate 5-HT receptor agonist

A3778 RS 127445 5-HT2B receptor antagonist,high affinity

A3697 Palonosetron 5-HT3 antagonist

A3157 Alosetron 5-HT3 receptor antagonist

A3158 Alosetron (Z)-2-butenedioate 5-HT3 receptor antagonist

A3159 Alosetron Hydrochloride 5-HT3 receptor antagonist,potent and highly selective

A3160 Alosetron Hydrochloride(1:X) 5-HT3 receptor antagonist

A3192 Asenapine hydrochloride Atypical antipsychotic

A3239 B-HT 920 D2 receptor agonist

A3241 Bilobalide Neuroprotective agent

A3317 Clozapine N-oxide (CNO) Metabolite of clozapine, used in chemogenetics.

A3330 CP-809101 5-HT2C receptor agonist

A3331 CP-809101 hydrochloride 5-HT2C receptor agonist, potent and selective

A3443 Granisetron Serotonin 5-HT3 receptor antagonist

A3569 LY 344864 5-HT1F receptor agonist,potent and selective

A5010 Asenapine Inhibits adrenergic receptor/5-HT receptor

B1001 Loxapine 5-HT receptor antagonist

B2265 BRL-15572 5-HT1D receptor antagonist

B2245 BRL-54443 5-HT1E/1F receptor agonist,potent and selective

B1198 Cisapride 5-HT4 receptor agonist

B2256 SB742457 5-HT6 receptor antagonist,highly selective and high affinity

B2240 Olanzapine Antagonist of 5-HT2A and dopamine D2 receptors

B1199 Tandospirone Anxiolytic and antidepressant reagent

B1058 Lasmiditan 5-HT1F receptor agonist

B2254 SB269970 HCl 5-HT7 receptor antagonist,potent and selective

B1200 PRX-08066 5-HT2BR antagonist

B2262 Agomelatine MT1/MT2 / 5-HT2C agonist

B1201 Agomelatine hydrochloride Norepinephrine-dopamine disinhibitor (NDDI)

B1202 Agomelatine L(+)-Tartaric acid Norepinephrine-dopamine disinhibitor (NDDI)

B1197 Risperidone mesylate 5-HT2 receptor blocker

B1196 Risperidone hydrochloride 5-HT2 receptor blocker

A2436 Fluoxetine HCl Serotonin reuptake inhibitor,selective

A2553 Fluvoxamine maleate Serotonin reuptake inhibitor,selective,antidepressant

A5355 Venlafaxine Dual serotonin/noradrenalin re-uptake inhibitor

A5322 Tianeptine sodium 5-HT uptake facilitator,selective,antidepressant

A5294 Sumatriptan Succinate 5-HT1 receptor agonist

A5350 Ziprasidone HCl Serotonin and dopamine receptor antagonist

A5399 Iloperidone Dopamine (D2) and serotonin (5HT2) receptor antagonist

A2547 Vortioxetine (Lu AA21004) HBr 5-HT receptor modulator, antidepressant and anxiolytic

A2098 PRX-08066 Maleic acid 5-HT2B receptor antagonist,potent and selective

A8514 Risperidone SR-2A inhibitor

A8516 Rizatriptan Benzoate 5-HT Receptor agonist

A8384 Blonanserin Atypical antipsychotic

A8421 Duloxetine HCl 5-HT receptor inhibitor

C4117 Imipramine (hydrochloride) serotonin and norepinephrine transporters inhibitor

C4077 Nortriptyline (hydrochloride) norepinephrine and serotonin transporters blocker

B7848 RS 127445 HCl 5-HT2B receptor antagonist,high affinity

C5214 6-fluoro-DL-Tryptophan serotonin (5-HT) synthesis inhibitor

C5271 AL 34662 potent 5-HT2 receptor agonist

B4981 Sumatriptan 5-HT1 receptor agonist

A5166 Ondansetron HCl 5-HT3 receptor antagonist

A3793 SB 271046 hydrochloride Selective 5-HT6 antagonist

A3777 Rotigotine hydrochloride Agonist of dopamine D2/D3 receptor

A3776 Rotigotine Agonist of dopamine D2/D3 receptor

A3748 rac-Rotigotine Hydrochloride Agonist of dopamine D2/D3 receptor

A3561 Lu AE58054 Hydrochloride 5-HT(6)R antagonist

A3560 Lu AE58054 5-HT(6)R antagonist

C5582 3,4-dihydro Naratriptan selective serotonin 5-HT1B agonist

Product Name	5-HTR	5-HT1R	5-HT1AR	5-HT1BR	5-HT1DR	5-HT1FR	5-HT2R	5-HT2AR	5-HT2BR	5-HT2CR	5-HT3R	5-HT3AR	5-HT4R	5-HT5AR	5-HT6R	5-HT7R	5-HT uptake	Other Targets
Palonosetron											*
Palonosetron HCl											*
Ondansetron hydrochloride dihydrate											*
Tropisetron Hydrochloride											***							α7-nicotinic receptor (agonist)
Tropisetron											***							α7-nicotinic receptor (agonist)
Lurasidone HCl			****					****								*****		Dopamine D2 noradrenaline α2C
Pizotifen	*
Iloperidone hydrochloride							*											Dopamine D2
SB-269970																****
SB269970 HCl																****
PRX-08066									****
Agomelatine									**	**								melatonin receptors
Agomelatine hydrochloride									**	**
Agomelatine L(+)-Tartaric acid										*
Loxapine	*																	D2DR D4DR
Pizotifen Malate	*
Azasetron HCl											****
Ondansetron											*
Trazodone HCl	*
Clomipramine HCl																	*
Dapoxetine HCl																	*
Ketanserin								*
VUF 10166												*****
Amitriptyline HCl							**						****					serotonin receptor norepinephrine receptor sigma 1 receptor
Desvenlafaxine																	***	norepinephrine (NE) reuptake
Desvenlafaxine Succinate																	***	norepinephrine (NE) reuptake
LY310762					**
SB271046															****
Olanzapine							*											D2 dopamine receptor
SB 271046 hydrochloride			**	**	**	*									*****			D3
Vilazodone																	*
Vilazodone Hydrochloride																	*
Vortioxetine			***	***								****				***		SERT
WAY-100635 maleate salt			****
Granisetron											*
Granisetron HCl											*
Alosetron											*
Alosetron (Z)-2-butenedioate											*
Alosetron Hydrochloride(1:X)											*
Alosetron Hydrochloride											*
Asenapine hydrochloride			****	****				*****	*****	*****				****	*****	*****		adrenergic α1 (8.9) α2A (8.9) α2B (9.5) and α2C (8.9) receptors dopamine D1 (8.9) D2 (8.9) D3 (9.4) and D4 (9.0) histamine H1 (9.0) and H2 (8.2) receptors.
Asenapine			****	****				*****	*****	*****				****	*****	*****		adrenergic α1 (8.9) α2A (8.9) α2B (9.5) and α2C (8.9) receptors dopamine D1 (8.9) D2 (8.9) D3 (9.4) and D4 (9.0) histamine H1 (9.0) and H2 (8.2) receptors.
Clozapine N-oxide							*
Lu AE58054															*****
Lu AE58054 Hydrochloride															*****
Mosapride											*
Mosapride Citrate											*
Fluoxetine HCl																	*****
Blonanserin							*											D2 receptor
Duloxetine HCl																	*
Risperidone hydrochloride							*****											dopamine D2 receptor
Risperidone mesylate							*****											dopamine D2 receptor
Risperidone							*****											dopamine D2 receptor
BRL-15572			***		***			**	***							**
SB742457															*****
PRX-08066 Maleic acid									****
Fluvoxamine maleate	****																*
Ondansetron HCl											*
Ziprasidone HCl			****		****			*****		****								dopamine receptor
Iloperidone							*											dopamine receptor
Vortioxetine (Lu AA21004) HBr			***	***								****				***		SERT
LY 393558				*****	****			***	***								****
BGC 20-761															***
NPS ALX Compound 4a dihydrochloride															*****
SB 399885 hydrochloride															*****
SGS 518 oxalate															*
Zotepine								*****										dopamine D2 receptor histamine H1 receptor
LY 266097 hydrochloride									*****
MDL 100907								*****
SB 699551														****
Melperone hydrochloride								**										D2 receptor adrenergic α1/α2 receptors
Fananserin			***					*****										dopamine D4 histamine H1 adrenergic α1 D2 receptors
Amperozide hydrochloride							***
Nefazodone hydrochloride								****										serotonin and noradrenalin uptake
Ro 04-6790															***
1-Methylpsilocin									***
LY 272015 hydrochloride								***	*****	***
LY 334370 hydrochloride			***			****
SB 258719 hydrochloride																*
SB 242084										*
SB 243213 dihydrochloride								**	***	*****
MS 245 oxalate															****
AT 1015								*
EMD 281014 hydrochloride								*****		**
DV 7028 hydrochloride							***
S 32212 hydrochloride										****
PU 02												**
SB 200646 hydrochloride								*	***	**
R 1485 dihydrochloride															****
DR 4485 hydrochloride																****
SB 203186 hydrochloride													*
RS 39604 hydrochloride													*****
Methysergide maleate		*					*
Methylergometrine maleate		*					*
Metergoline		*			*		*								*	*
3-AQC											*
RS 23597-190 hydrochloride													*
2-[1-(4-Piperonyl)piperazinyl]benzothiazole											*
MDL 11,939								****
N-Desmethylclozapine										*
4F 4PP oxalate								****
Cinanserin hydrochloride							*
Methiothepin maleate		*					*
MDL 72222											*
Spiperone hydrochloride								*
PNU 109291					*
SB 204070													*****
GR 55562 dihydrochloride				***	**
SB 206553 hydrochloride									****	***
R-96544 hydrochloride							****	****
Zacopride hydrochloride											*****
Altanserin hydrochloride			*					*****		***								adrenergic α1 receptors dopamine D2 receptors
Ritanserin							*****
SB 258585 hydrochloride															****
SDZ 205-557 hydrochloride											*		*
GR 125487 sulfamate													*****
Mesulergine hydrochloride								*****		*****								D2-like dopamine receptor
LY 215840							*									*
SB 224289 hydrochloride				****
SB 216641 hydrochloride				*
SDZ SER 082 fumarate			*						*	*
GR 113808													*****
SB 204741									***	*
SB 228357								***	****	*****
SB 221284								**	***	****
NAS-181				***
GR 127935 hydrochloride				****	****
Pimavanserin								****
Dihydroergotamine mesylate	*																	adrenergic α receptors dopamine D2 receptors (Agonist)
Sarpogrelate hydrochloride								****	**	***
Ramosetron Hydrochloride											*
Eltoprazine			***	***						***
Eltoprazine hydrochloride			***	***						***
Fluvoxamine																	*
Citalopram hydrobromide																	****
Indatraline hydrochloride																	*****	dopamine (DAT) and noradrenalin (NET) uptake
Paroxetine maleate																	*****
(±)-McN 5652																	*****	noradrenalin and dopamine uptake
Lofepramine																	*	noradrenalin re-uptake
BTS 54-505 hydrochloride																	*	noradrenalin re-uptake
NAD 299 hydrochloride			*****
WY 45233 succinate																	***
Dexfenfluramine hydrochloride																	*
(S)-WAY 100135 dihydrochloride			***
Cyanopindolol hemifumarate			*	*														β-adrenoceptor
Ketanserin								*
MDL 73005EF hydrochloride			*
MDL 72832 hydrochloride			*
NAN-190 hydrobromide			*
CGS 12066B dimaleate				*
Anpirtoline hydrochloride											***
MM 77 dihydrochloride			*
Isamoltane hemifumarate				*														β-adrenergic receptors
(±)-MDMA hydrochloride																	*	dopamine uptake
WAY-100635			****
Ziprasidone			****		****			*****		****
Ziprasidone hydrochloride monohydrate			****		****			*****		****
RS 127445									*****
B-HT 920											*							Dopamine D2 receptor α2-adrenoceptor (agonist)
Clozapine N-oxide	*
Venlafaxine																	*	noradrenalin re-uptake

Product Name	5-HTR	5-HT1R	5-HT1AR	5-HT1BR	5-HT1CR	5-HT1DR	5-HT1ER	5-HT1FR	5-HT2R	5-HT2AR	5-HT2BR	5-HT2CR	5-HT2HR	5-HT3R	5-HT4R	5-HT4AR	5-HT4BR	5-HT6R	5-HT7R	5-HT uptake	Other Targets
Tandospirone			***
Eletriptan HBr				*		*
Lasmiditan								****
Lorcaserin HCl												***
Mosapride															*
Mosapride Citrate															*
Naratriptan		*
Almotriptan Malate				*		*
Urapidil HCl			*																		α1-adrenoceptor(antagonist)
WAY-100635 Maleate			****
Zolmitriptan	*
BMY 7378		****																			α2C-adrenoceptor α1D-adrenoceptor
Prucalopride																****	****
CP 93129 dihydrochloride				****
Adoprazine			*																		D2/3 receptor (antagonist)
Tianeptine																				*
Tianeptine sodium																				***
Vilazodone			*
Vilazodone Hydrochloride			*
Rotigotine hydrochloride			*																		dopamine D2 D3 receptor adrenergic α2B receptors
Rotigotine			*																		dopamine D2 D3 receptor adrenergic α2B receptors
rac-Rotigotine Hydrochloride			*																		dopamine D2 D3 receptor adrenergic α2B receptors
CP-809101										**	***	*****
CP-809101 hydrochloride										**	***	*****
Mosapride Citrate															*
BRL-54443							****	****
Cisapride															*
Rizatriptan Benzoate						*
ML 10302 hydrochloride														**	****
Org 12962 hydrochloride										**	**	***
Donitriptan hydrochloride				*****		*****
CP 135807						*
NPEC-caged-serotonin	*
CJ 033466															*****
LP 44																			*****
TCB-2										*****
L-703,664 succinate			**			***
LP 12 hydrochloride			***							**									*****		dopamine D2 receptors
1-Methylpsilocin										**		***
EMD 386088 hydrochloride														***				****
EMDT oxalate																		***
LP 20 hydrochloride			**																****
Org 37684										***	***	****
DOB hydrochloride													*****
DOI hydrochloride										*****	*	****
ST 1936 oxalate																		***
BIMU 8															***
Tegaserod maleate															***
NBOH-2C-CN hydrochloride										****
2-Methyl-5-hydroxytryptamine hydrochloride														*				***
GR 46611						*
RS 67333 hydrochloride															****
Psilocin	*
m-Chlorophenylbiguanide hydrochloride														*
α-Methyl-5-hydroxytryptamine maleate										**	****	***
2-[1-(4-Piperonyl)piperazinyl]benzothiazole															*
L-694,247						*
MK 212 hydrochloride										**		***
RS 56812 hydrochloride														*****
RS 67506 hydrochloride															****
N-Methylquipazine dimaleate														*
Quipazine dimaleate														*
1-Phenylbiguanide hydrochloride														*
PNU 142633						****
WAY 208466 dihydrochloride																		****
m-CPP hydrochloride										**	***	***
5-Carboxamidotryptamine maleate		*
Zacopride hydrochloride															**
WAY 161503 hydrochloride												****
Ro 60-0175 fumarate												*
AS 19																			*****
WAY 629 hydrochloride										*		***						*	**
PNU 22394 hydrochloride										***	***	***
BW 723C86 hydrochloride											*
SR 57227 hydrochloride														*
CP 94253 hydrochloride			***	****	**	***			*
S 14506 hydrochloride			*****	**	***				**					*
Ipsapirone			****
(R)-(+)-8-Hydroxy-DPAT hydrobromide			*
MDL 72832 hydrochloride			*
8-Hydroxy-DPAT hydrobromide			*																**
BP 554 maleate			*
Anpirtoline hydrochloride			**	***					*
8-Hydroxy-PIPAT oxalate			*****
5-Nonyloxytryptamine oxalate				*****
LY 344864								****
Sumatriptan Succinate			***	***		***
Sumatriptan			***	***		***

Biochemicals