Potassium Channel
Potassium channels are voltage-gated ion channels that selectively permeate potassium ion through the excitable membrane. It regulates the release of neurotransmitters, insulin secretion, smooth muscle contraction and heart rate etc.
- B2193 Mitiglinide CalciumTarget: Inward Rectifier Potassium (Kir) ChannelsSummary: Potassium channel inhibitor
- B2194 TolbutamideTarget: cAMP|Sulfonylurea receptorsSummary: first generation potassium channel blocker
- B2195 GliclazideTarget: Inward Rectifier Potassium (Kir) ChannelsSummary: Potassium channel inhibitor
- B2198 NateglinideTarget: Inward Rectifier Potassium (Kir) ChannelsSummary: Insulin secretagog agent
- B4849 AzimilideSummary: class III anti-arrhythmic drug
- B6591 IberiotoxinSummary: blocker of the big conductance Ca2+-activated K+ channel
- B7388 ValinomycinTarget: IonophoresSummary: potassium-specific transporter
- B7659 Psora 41 CitationTarget: Voltage-gated Potassium (KV) ChannelsSummary: Kv1.3 blocker
- A1888 TRAM-34Target: Calcium-Activated Potassium (KCa) ChannelsSummary: KCa3.1 blocker,potent and highly selective