Leukotriene Receptor
Leukotrienes receptors are divided into two types, BLT receptors and CycLT receptors. BLT receptors mediate chemoattraction. CysLT receptors mediate pro-inflammatory effects including constriction of airways ad smooth muscle contraction.
- B6999 FPL 55712Summary: Leukotriene receptor antagonist
- B7011 Leukotriene B4Summary: BLT1/BLT2 receptor agonist
- B7023 MK-571Target: Leukotriene and Related ReceptorsSummary: leukotriene D4 receptor antagonist, orally active
- B7284 BAY-u 9773Summary: Antagonist of CysLT1/CysLT2 receptors
- B6860 SR 2640 hydrochlorideSummary: leukotriene D4 and E4 receptor antagonist
- B6930 CinalukastSummary: CysLT1 (LTD4) leukotriene receptor antagonist
- B6978 LY 255283Summary: BLT2 receptor antagonist