Leukotriene Receptor
Leukotrienes receptors are divided into two types, BLT receptors and CycLT receptors. BLT receptors mediate chemoattraction. CysLT receptors mediate pro-inflammatory effects including constriction of airways ad smooth muscle contraction.
- B6860 SR 2640 hydrochlorideSummary: leukotriene D4 and E4 receptor antagonist
- B6930 CinalukastSummary: CysLT1 (LTD4) leukotriene receptor antagonist
- B6978 LY 255283Summary: BLT2 receptor antagonist
- B2068 ZafirlukastTarget: Leukotriene and Related ReceptorsSummary: oral leukotriene receptor antagonist
- C5226 γ-Linolenic Acid methyl esterSummary: weak leukotriene B4 (LTB4) receptor antagonist
- C5416 REV 5901Summary: antagonist of cysteinyl-leukotriene receptors
- C5518 γ-Linolenic AcidSummary: weak LTB4 receptor antagonist