Adrenergic Receptor
Adrenergic receptor is a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.
- C3067 Niguldipine (hydrochloride)Summary: α1A-adrenoceptor antagonist
- C3965 Rilmenidine (hemifumarate)Summary: I1-imidazoline binding site selective ligand and α2-adrenoceptor agonist
- C3990 Lofexidine (hydrochloride)Summary: α2-adrenergic receptor agonist
- C3786 Guanabenz (hydrochloride)Summary: α2-adrenergic receptor agonist
- C3632 ZilpaterolSummary: β-adrenergic receptor agonist
- C4034 (±)-4-hydroxy Propranolol (hydrochloride)Summary: β1- and β2-adrenergic receptors inhibitor
- C4493 Midodrine (hydrochloride)Summary: prodrug of the α1-adrenergic receptor agonist
- C3003 (±)-TalinololSummary: β1-selective adrenoceptor antagonist
- C3031 (R)-(+)-AtenololSummary: less active enantiomer of the racemic β1-adrenergic receptor antagonist, (R,S)-atenolol.
- C4521 Celiprolol (hydrochloride)Summary: β1 adrenergic receptor antagonist and β2 adrenergic receptor partial agonist