ATM/ATR
ATM (ataxia telangiectasia mutated) and ATR (ATM- and Rad3-related) are two PIKKs (phosphatidylinositol 3-kinase-like kinases) that regulate the DNA damage response (DDR) pathways.
- A3210 AZ201 CitationTarget: ATM/ATRSummary: ATR inhibitor,potent and selective
- A8336 KU-600192 CitationTarget: ATM/ATRSummary: ATM kinase inhibitor,potent and selective
- A8626 ETP-46464Target: PI3K|mTOR|DNA-PK|ATM/ATRSummary: ATR inhibitor,potent and selective
- B1383 VE-8222 CitationTarget: ATM/ATRSummary: ATR inhibitor