Biochemical Reagent
- BA5511 CycrimineSummary: Cycrimine is an orally active muscarinic cholinergic receptor antagonist that reduces acetylcholine levels in a Parkinson's model.
- BA5512 TBPBSummary: TBPB is an M1mAChR variant agonist.
- BA5513 JHU37152Summary: JHU37152 is a potent and permeable agonist across the blood-brain barrier.
- BA5514 ML375Summary: ML375 (VU0483253) is a potent, highly selective, blood-brain-barrier-crossing and orally active negative-alteration modulator (NAM) with M5's of 300 nM and 790 nM for human and rat, respectively.
- BA5515 ArborineSummary: Inhibits the peripheral effects of acetylcholine and induces a fall in blood pressure.
- BA5516 AnisodamineSummary: Anisodamine (6-Hydroxyhyoscyamine), belladonna alkaloid, is also a non-subtype-selective muscarinic and nicotinic cholinergic receptor antagonist.
- BA5517 AC260584Summary: AC260584 is a muscarinic receptor variant agonist.
- BA5518 ML381Summary: ML381 (VU0488130) is a highly selective
- BA5519 FesoterodineSummary: Fesoterodine is an orally effective, non-subtype-selective, competitive muscarinic receptor antagonist.
- BA5520 ZamifenacinSummary: Zamifenacin (UK-76654) is a potent intestinal selective muscarinic receptor antagonist.