Bioactive Compounds
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A5057 MGCD-265 analogTarget: VEGFR|c-METSummary: Met/Flt/Flk/Ron/Tie-2 inhibitor -
A5449 PIK-93Summary: PI3Kγ/PI4KIIIβ/PI3Kα inhibitor -
A5455 AEE788 (NVP-AEE788)Summary: EGFR/HER-2/VEGFR inhibitor -
A5511 OfloxacinTarget: Topoisomerases|DNA gyraseSummary: Fluoroquinolones,antibiotics -
A5719 AT7519Target: Cyclin-Dependent KinasesSummary: Multi-CDK inhibitor -
A1947 MEK162 (ARRY-162, ARRY-438162)Target: MEKSummary: MEK1/2 inhibitor,potent and selective -
A8331 Bleomycin Sulfate13 CitationSummary: DNA synthesis inhibitor -
A8460 LevodopaSummary: Dopamine precursor. -
A8413 Diperodon HClSummary: A prodrug compound activated by serum enzyme catalysis. -
B1583 UNC19993 CitationTarget: EZH2|EZH1Summary: EZH2 inhibitor

