Bioactive Compounds
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B4763 GKT1378318 CitationTarget: NADPH OxidasesSummary: dual NADPH oxidase Nox1/Nox4 inhibitor -
B7784 AL 8697Target: p38Summary: p38α inhibitor,potent and selective -
B4846 LB-100Summary: protein phosphatase 2A(PP2A)inhibitor -
B4917 Ischemin sodium saltSummary: CBP bromodomain inhibitor -
B4920 EC 144Target: HSP90Summary: High affinity, potent and selective Hsp90 inhibitor -
B5859 EntrectinibTarget: Trk Receptors|ALK|ROS1Summary: Orally active inhibitor of ALK kinase -
B5942 AS601245Summary: c-Jun NH2-terminal protein kinase inhibitor -
A1044 Gap 2624 CitationTarget: Gap JunctionsSummary: Gap junction blocker peptide, mapping to connexin 43 residue 63-75 -
A8737 S6384540 CitationTarget: MCL1Summary: MCL1 inhibitor -
B1173 B-Raf inhibitor 1 dihydrochlorideSummary: B-Raf inhibitor,potent and selective
