Bioactive Compounds
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B4825 IKKε-IN-1Summary: potent IKKε inhibitor -
B4918 OXF BD 02Summary: Selective inhibitor of the first bromodomain of BRD4 -
B4937 SB 706504Summary: p38 MAPK inhibitor -
A8715 SBI-02069658 CitationTarget: ULK1Summary: ULK1 inhibitor -
B5904 Regadenoson1 CitationTarget: Adenosine A2A ReceptorsSummary: Highly selective and low affinity A2A adenosine agonist -
B5960 PF-03394197(Oclacitinib)Summary: Novel Janus kinase inhibitor -
B5970 Sanguinarine chlorideSummary: Inhibitor of PP2C and MKP-1 -
A1045 Gap 279 CitationTarget: Gap JunctionsSummary: Selective gap junction blocker -
B2117 Pioglitazone1 CitationSummary: PPAR agonist -
B1407 Dabrafenib (GSK2118436)3 CitationTarget: RafSummary: Inhibitor of BRAF(V600) mutants

