EGFR
- A8322 Neratinib (HKI-272)3 CitationTarget: EGFRSummary: HER2/EGFR inhibitor,potent and irreversible
- A8319 Dacomitinib (PF299804, PF299)Target: ErbBSummary: HER inhibitor
- A8247 Afatinib (BIBW2992)1 CitationTarget: EGFRSummary: Irreversible EGFR/HER2 inhibitor
- A8234 Erlotinib Hydrochloride2 CitationSummary: Selective EGFR inhibitor
- A8219 Gefitinib (ZD1839)15 CitationTarget: EGFRSummary: Selective EGFR inhibitor
- A8218 Lapatinib7 CitationTarget: ErbBSummary: EGFR/HER2 inhibitor,potent,selective and reversible
- A8199 PD153035 hydrochloride1 CitationTarget: EGFRSummary: Potent EGFR inhibitor
- A8197 Compound 561 CitationTarget: EGFRSummary: REGFR inhibitor
- A5455 AEE788 (NVP-AEE788)Summary: EGFR/HER-2/VEGFR inhibitor
- A4139 AG-4903 CitationTarget: EGFR|JAKSummary: JAK2/EGFR inhibitor