EGFR
- A2689 ButeinTarget: Src|STAT|EGFR|Angiotensin-Converting Enzymes (ACEs)|5-Lipoxygenases|PTK|enoyl-acyl-carrier protein reductaseSummary: Protein kinase inhibitor
- A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: HER2 inhibitor,potent and selective
- A2024 PD168393Target: PDGFR|FGFR|EGFR|PKC|insulinSummary: EGFR inhibitor
- A1845 Canertinib (CI-1033)Summary: HER family tyrosine kinase inhibitor
- A1835 Pelitinib (EKB-569)Summary: EGFR inhibitor,potent and irreversible
- A1393 WZ8040Target: EGFRSummary: EGFR T790M inhibitor,irreversible amd potent
- A1389 WZ4002Summary: Mutant-selective EGFR inhibitor(L858R,T790M), irreversible and potent
- A1367 ALK-IN-1Summary: Anaplastic lymphoma kinase (ALK) inhibitor
- A1173 AG-18Summary: EGFR/PDGFR inhibitor