EGFR
- B1104 AZD-92911 CitationTarget: EGFRSummary: Mutated forms EGFR inhibitor
- B1103 Mutant EGFR inhibitorSummary: Selective Mutated EGFR inhibitor
- B1020 AST-1306 TsOHSummary: ErbB2 and EGFR inhibitor
- A8881 WZ3146Summary: Mutant EGFR inhibitor, potent and irreversible
- A8696 FIIN-2Target: FGFRSummary: Irreversible inhibitor of FGFR
- A8375 AZD8931 (Sapitinib)Target: EGFR|ErbBSummary: ErbB inhibitor
- A8367 AST-1306Summary: EGFR/HER2 inhibitor
- A8366 ARRY-380Target: HER2Summary: Tyrosine kinase HER2 and p95-HER2 inhibitor
- A8365 Varlitinib (ARRY334543)Summary: ErbB inhibitor
- A8357 AG-1478Target: EGFRSummary: EGFR inhibitor,potent and selective