Takinib
Catalog No.
BA2736
Takinib (EDHS-206) is a potent and selective inhibitor (=9.5nM)
Featured Products
Takinib (EDHS-206) is a potent and selective inhibitor (=9.5nM), acting 1.5log-fold more potently than (=120nM) and (=390nM).Takinib is an inhibitor of TAK1 autophosphorylation and binds non-competitively within the ATP-binding pocket. Takinib induced TNF-α-stimulated apoptosis in rheumatoid arthritis and metastatic breast cancer cell models.Takinib is also an inhibitor of Plasmodium falciparum protein kinase 9 (Kof0.46nM).
| Physical Appearance | A solid |
| Storage | -20°C |
| M.Wt | 322.36 |
| Cas No. | 1111556-37-6 |
| Formula | C18H18N4O2 |
| Synonyms | EDHS-206 |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |