Signaling Pathways
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A2521 VE-8212 CitationSummary: ATR kinase inhibitor -
A2477 Tyrphostin AG 12961 CitationTarget: PDGFRSummary: PDGFR inhibitor,selective and ATP-competitive -
A2623 VU 0364439Summary: Positive allosteric mGluR-4 modulator -
A1174 AMG-517Target: TRP ChannelSummary: TRPV1 antagonist,potent and highly selective -
A1387 AZD53636 CitationTarget: AktSummary: AKT inhibitor,pyrrolopyrimidine derived -
A2689 ButeinTarget: Src|STAT|EGFR|Angiotensin-Converting Enzymes (ACEs)|5-Lipoxygenases|PTK|enoyl-acyl-carrier protein reductaseSummary: Protein kinase inhibitor -
A1413 CEP-32496Summary: BRAF(V600E)inhibitor,highly potent -
A1929 MacitentanSummary: Endothelin (ET)(A) and ET(B) receptor antagonist -
A2173 SC 1441 CitationTarget: GlycoproteinsSummary: Gp130 inhibitor -
A2005 Nutlin-3bTarget: p53-MDM2 interactionSummary: MDM2/p53 inhibitor

