Relugolix
Catalog No.
BA5360
Relugolix (TAK-385) is a potent, orally active, nonpeptide gonadotropin-releasing hormone antagonist.
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Relugolix (TAK-385) is a potent, orally active, non-peptide gonadotropin-releasing hormone antagonist. Relugolix has high affinity and strong antagonistic activity for human (=0.33 nM) and monkey (=0.32 nM) receptors compared to TAK-013 (HY-100209).Relugolix is used in the study of sex hormone-dependent diseases such as endometriosis, uterine fibroids, and prostate cancer.
| Physical Appearance | A solid |
| Storage | -20°C |
| M.Wt | 623.63 |
| Cas No. | 737789-87-6 |
| Formula | C29H27F2N7O5S |
| Synonyms | TAK-385 |
| Solubility | ≥50.9 mg/mL in DMSO; insoluble in EtOH; insoluble in H2O |
| Chemical Name | 1-(4-(1-(2,6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-3-methoxyurea |
| Canonical SMILES | O=C(NOC)NC1=CC=C(C(S2)=C(CN(C)C)C(C(N3C4=NN=C(OC)C=C4)=O)=C2N(CC5=C(F)C=CC=C5F)C3=O)C=C1 |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |
Quality Control & MSDS
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Chemical structure
