Razuprotafib
Catalog No.
BA8081
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Razuprotafib (AKB-9778) is a potent and selective inhibitor of catalytic activity (=17pM) that promotes TIE2 activation, enhances ANG1-induced TIE2 activation, and stimulates phosphorylation of signaling molecules in the TIE2 pathway, including AKT, eNOS, and .Razuprotafib inhibits the structure-associated phosphatase PTP1B with an IC of 780 nM.Razuprotafib has good selectivity for VE-PTP except for HPTPη (IC=36 pM) and HPTPγ (100 pM).
| Physical Appearance | A solid |
| Storage | -20°C |
| M.Wt | 586.70 |
| Cas No. | 1008510-37-9 |
| Formula | C26H26N4O6S3 |
| Synonyms | AKB-9778 |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |