Metarrestin
Catalog No.
BA3987
Metarrestin (ML246) is an orally effective, first-in-class, selective perinuclear compartment inhibitor.
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Metarrestin (ML246) is an orally potent, first-in-class, selective inhibitor of perinuclear compartmentalization.Metarrestin disrupts nucleolus structure and inhibits transcription, in part due to an interaction with the translation elongation factor eEF1A2.Metarrestin blocks metastatic progression and prolongs survival in a mouse cancer model.
| Physical Appearance | A solid |
| Storage | -20°C |
| M.Wt | 474.60 |
| Cas No. | 1443414-10-5 |
| Formula | C31H30N4O |
| Synonyms | ML246 |
| Solubility | ≥17.1 mg/mL in DMSO; ≥3.52 mg/mL in EtOH with ultrasonic; insoluble in H2O |
| Chemical Name | (1r,4r)-4-(7-benzyl-4-imino-5,6-diphenyl-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-3-yl)cyclohexan-1-ol |
| Canonical SMILES | N=C1N([C@H]2CC[C@H](O)CC2)C=NC3=C1C(C4=CC=CC=C4)=C(C5=CC=CC=C5)N3CC6=CC=CC=C6 |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |
Quality Control & MSDS
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Chemical structure
