Lumateperone
Catalog No.
BA5040
Lumateperone (ITI-007) is an orally active receptor antagonist (Ki=0.54nM)
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Lumateperone (ITI-007) is an orally active receptor antagonist (Ki=0.54nM), partial agonist at presynaptic D2 receptors and antagonist at postsynaptic D2 receptors (Ki=32nM), and modulator of the dopamine D1 receptor.Lumateperone has anticancer activity, and has been used in studies of schizophrenia and bipolar depression. Lumateperone has anticancer activity and is also used to study schizophrenia and bipolar depression.
| Physical Appearance | An oil |
| Storage | 4°C, protect from light |
| M.Wt | 393.50 |
| Cas No. | 313368-91-1 |
| Formula | C24H28FN3O |
| Synonyms | ITI-007 |
| Solubility | ≥50.6 mg/mL in DMSO; ≥25.05 mg/mL in EtOH; insoluble in H2O |
| Chemical Name | 1-(4-fluorophenyl)-4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)butan-1-one |
| Canonical SMILES | CN1C2=C3C([C@@]4([H])[C@@](CCN(C4)CCCC(C5=CC=C(C=C5)F)=O)([H])N3CC1)=CC=C2 |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |
Quality Control & MSDS
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Chemical structure
