Irdabisant
Catalog No.
BA5424
Irdabisant (CEP-26401) is a selective, orally active and blood-brain barrier permeable histamine H3 receptor (,H3R) antagonist/inverse agonist with 7.2 nM and 2.0 nM for rat H3R and human H3R, respectively.
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Irdabisant (CEP-26401) is a selective, orally active, and blood-brain barrier permeable histamine H3 receptor (,H3R) antagonist/inverse agonist with 7.2 nM and 2.0 nM for rat H3R and human H3R, respectively.Irdabisant has a relatively low inhibitory activity on hERG currents with an IC of 13.8 μM. Irdabisant has cognitive enhancement and arousal effects in a rat social cognitive model.Irdabisant can be used in studies of schizophrenia or cognitive disorders.
Physical Appearance | A solid |
Storage | -20°C |
M.Wt | 313.39 |
Cas No. | 1005402-19-6 |
Formula | C18H23N3O2 |
Synonyms | CEP-26401 |
Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
General tips | We do not recommend long-term storage for the solution, please use it up soon. |