GNE-0439
Catalog No.
BA6992
GNE-0439 is a novel selective inhibitor.
Featured Products
GNE-0439 is a novel selective inhibitor of Nav1.5 with a value of 0.34 uM and inhibits Nav1.5 with a value of 38.3 μM.GNE-0439 inhibits the mutant N1742K channel in a membrane potential assay (=0.37 uM).GNE-0439 has a carboxylic acid moiety that binds outside the channel pore, in contrast to the known selective VSD4 binders.
| Physical Appearance | A solid |
| Storage | Tightly sealed and desiccated at 4°C |
| M.Wt | 345.48 |
| Cas No. | 1241902-40-8 |
| Formula | C21H31NO3 |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |