Ensifentrine
Catalog No.
BA8157
Ensifentrine (RPL-554) is an inhaled, first-of-its-kind phosphodiesterase 3 and dual inhibitor of 0.4nM and 1479nM, respectively.
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Ensifentrine (RPL-554) is an inhaled, first-in-class phosphodiesterase 3 and dual inhibitor at 0.4 nM and 1479 nM, respectively.Ensifentrine has bronchoprotective and anti-inflammatory activity and may be used in chronic obstructive pulmonary disease (COPD) studies.
| Physical Appearance | A solid |
| Storage | -20°C |
| M.Wt | 477.56 |
| Cas No. | 1884461-72-6 |
| Formula | C26H31N5O4 |
| Synonyms | RPL-554 |
| Solubility | ≥8.67 mg/mL in DMSO; insoluble in EtOH; insoluble in H2O |
| Chemical Name | (E)-1-(2-(2-(mesitylimino)-9,10-dimethoxy-4-oxo-6,7-dihydro-2H-pyrimido[6,1-a]isoquinolin-3(4H)-yl)ethyl)urea |
| Canonical SMILES | O=C(NCCN1C(N(C2=C/C1=N\C3=C(C=C(C=C3C)C)C)CCC4=C2C=C(C(OC)=C4)OC)=O)N |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |
Quality Control & MSDS
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Chemical structure
