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EED226

Catalog No.
BA4812
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EED226, a multi-comb inhibitor of complex 2, binds to the K27me3 pocket on embryonic ectodermal development (EED) and exhibits potent antitumor activity in a transplanted tumor mouse model.
Grouped product items
SizePriceStock Qty
1mL(10 mM in DMSO)
$59.00
Ship with 10-15 days
5mg
$54.00
Ship with 10-15 days
10mg
$81.00
Ship with 10-15 days
25mg
$135.00
Ship with 10-15 days
50mg
$224.00
Ship with 10-15 days
100mg
$405.00
Ship with 10-15 days
For scientific research use only and should not be used for diagnostic or medical purposes.

Tel: +1-832-696-8203

Email: [email protected]

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Background

EED226, a multi-comb inhibitor of complex 2, binds to the K27me3 pocket on embryonic ectodermal development (EED) and exhibits potent antitumor activity in a mouse model of transplanted tumors.EED226 is a potent, orally bioavailable, selective EED inhibitor. When the H3K27me0 peptide was used as a substrate for an in vitro enzymatic assay, EED226 inhibited at a value of 23.4 nM.

Chemical Properties

Physical AppearanceA solid
Storage-20°C
M.Wt369.40
Cas No.2083627-02-3
FormulaC17H15N5O3S
Solubility≥51.3 mg/mL in DMSO; insoluble in EtOH; insoluble in H2O
Chemical NameN-(furan-2-ylmethyl)-8-(4-(methylsulfonyl)phenyl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
SDFDownload SDF
Canonical SMILESO=S(C1=CC=C(C2=CN=C(NCC3=CC=CO3)N4C2=NN=C4)C=C1)(C)=O
Shipping ConditionSmall Molecules with Blue Ice, Modified Nucleotides with Dry Ice.
General tips We do not recommend long-term storage for the solution, please use it up soon.