Darusentan
Catalog No.
BA5315
Darusentan (Lu-135252) is a selective endothelin receptor A receptor antagonist.
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Darusentan (Lu-135252) is a selective endothelin receptor A receptor antagonist with values of 1.4 nM with ET-A receptors and 184 nM with ET-B receptors, and more than 100-fold more selective for ETA receptors than for ETB receptors.Darusentan competes in the membranes of rat aortic vascular smooth muscle cells (RAVSMs) to binding of radiolabeled endothelin with a value of 13 nM.
| Physical Appearance | A solid |
| Storage | -20°C |
| M.Wt | 410.42 |
| Cas No. | 171714-84-4 |
| Formula | C22H22N2O6 |
| Synonyms | Lu-135252 |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |