CHMFL-PI3KD-317
Catalog No.
BA8770
CHMFL-PI3KD-317 is a potent, selective, and orally available inhibitor.
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CHMFL-PI3KD-317 is a potent, selective, orally available inhibitor with a value of 6 nM, which is 10-1500 times more selective than for other PIKK families such as (IC, 62.6 nM), (IC, 284 nM), (IC, 202.7 nM), PIK3C2A (IC, >10,000 nM), PIK3C2B (IC, 882.3nM), (IC, 1801.7nM), PI4KIIIA (IC, 574.1nM) and PI4KIIIB (IC, 300.2nM). In Raji cells, CHMFL-PI3KD-317 inhibited mediated T308 phosphorylation with an EC of 4.3 nM.CHMFL-PI3KD-317 had antiproliferative effects on cancer cells.
| Physical Appearance | A solid |
| Storage | -20°C |
| M.Wt | 494.03 |
| Cas No. | 2244992-76-3 |
| Formula | C21H24ClN5O3S2 |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |