Metabolic Enzyme/Protease
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BA4464 RG-12525Summary: RG-12525 is a specific, competitive, orally available antagonist. - BA4462 FK614Summary: FK614 is an orally active non-thiazolidinedione (TZD) type selective modulator.
- BA4459 BAY-5094Summary: BAY-5094 is an inverse agonist.
- BA4458 25-Hydroxytachysterol3Summary: 25-Hydroxytachysterol3 is the metabolite.
- BA4457 ConvallatoxinSummary: Convallatoxin is a cardiac glycoside isolated from RegeletRadde.
- BA4456 ST247Summary: ST247 is a potent inverse agonist.
- BA4455 BAY-5516Summary: BAY-5516 is an inverse agonist (6.1 ± 3.6 nM).
- BA4453 MavodelparSummary: Mavodelpar (REN001) is a selective agonist.
- BA4451 PTGR2-IN-1Summary: PTGR2-IN-1 is a potent inhibitor.
- BA4450 HWL-088Summary: HWL-088 is a potent, orally active free fatty acid receptor 1 agonist (at 18.9 nM) with moderate activity (at 570.9 nM).