Metabolic Enzyme/Protease
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C8954 Vardenafil hydrochlorideSummary: Vardenafil hydrochloride is a selective phosphodiesterase-5 inhibitor targeting cGMP signaling, widely utilized as a pharmacological probe in vascular and smooth muscle research. -
C8953 Menadione bisulfite sodiumSummary: Menadione bisulfite sodium is a water-soluble vitamin K3 derivative that modulates redox signaling and is widely utilized in oxidative stress and cell biology research. -
C8951 Efonidipine hydrochloride monoethanolateSummary: Efonidipine hydrochloride monoethanolate is a dual L- and T-type calcium channel blocker used as a pharmacological tool in cardiovascular signaling research. -
C8945 Eliglustat hemitartrateSummary: Eliglustat hemitartrate is a potent glucosylceramide synthase inhibitor targeting glycosphingolipid biosynthesis, widely utilized in sphingolipid metabolism and lysosomal pathway research. -
C8940 D-Gluconic acid (50% w/w in H2O)Summary: D-Gluconic acid (50% w/w in H2O) is a sugar acid metabolite used as a chelating and pH-modulating reagent in biochemical analysis, microbial metabolism, and enzymology research. -
C8927 Choline theophyllinateSummary: Oxtriphylline is a methylxanthine phosphodiesterase inhibitor and adenosine receptor antagonist used to investigate cyclic nucleotide signaling in pharmacological and biochemical research. -
C8920 Tofogliflozin(CSG 452)Summary: Tofogliflozin (CSG 452) is a potent, selective sodium-glucose cotransporter 2 inhibitor targeting renal glucose transport, widely utilized in metabolic and diabetes mechanism research. -
C8916 umbralisib (TGR-1202)Summary: Umbralisib (TGR-1202; CAS 1532533-67-7) is a selective PI3Kδ and casein kinase-1ε inhibitor used in oncology and signal transduction research. -
C8915 EliglustatSummary: Eliglustat is a potent glucosylceramide synthase inhibitor targeting glycosphingolipid biosynthesis, widely utilized in sphingolipid metabolism and lysosomal biology research. -
C8914 FursultiamineSummary: Fursultiamine is a lipophilic thiamine derivative used to investigate vitamin B1 metabolism, thiamine-dependent enzymatic pathways, and cellular bioenergetics in biochemical research.
