Bioactive Compounds
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A4487 WR 1065Summary: P53/p21waf-1/MDM2 activator -
A8218 Lapatinib7 CitationTarget: ErbBSummary: EGFR/HER2 inhibitor,potent,selective and reversible -
A8210 GDC-094120 CitationTarget: PI3KSummary: PI3K inhibitor,potent and selective -
A5059 EdaravoneSummary: A radical scavenger and antioxidant -
A5760 KRN 633Summary: VEGFR inhibitor,ATP-competitive -
A8335 Palbociclib (PD0332991) Isethionate1 CitationTarget: Cyclin-Dependent KinasesSummary: CDK4/6 inhibitor,highly selective -
A8437 Gemcitabine11 CitationSummary: inhibitor of DNA synthesis -
A8600 Tankyrase Inhibitors (TNKS) 22Summary: Tankyrase inhibitor -
B2184 GDC-0980 (RG7422)Summary: Class I PI3K inhibitor for PI3Kα/β/δ/γ -
B1621 TAK-733Target: MEKSummary: MEK allosteric site inhibitor
