Bioactive Compounds
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B2307 LGK-9744 CitationSummary: PORCN inhibitor,potent and specific -
B2282 KX2-3911 CitationSummary: Src inhibitor,highly selective -
B1011 Bafetinib (INNO-406)2 CitationSummary: Bcr-Abl/Lyn tyrosine kinase inhibitor -
B1498 I-BET-7624 CitationTarget: BromodomainsSummary: BET inhibitor,highly potent -
B2289 SB505124Summary: ALK4/ALK5/ALK7 inhibitor -
B5372 HU 308Summary: CB2-receptor agonist -
B5482 MRK 016Summary: GABAA receptor inverse agonist -
B5532 NPS 2390Target: Glutamate (Metabotropic) Group I ReceptorsSummary: group I mGlu antagonist -
B5567 SMER 3Summary: yeast SCF family E3 ubiquitin ligase (SCFMet30) inhibitor -
B5597 SEN 12333Summary: α7 nicotinic acetylcholine receptor (nAChR) agonist

