Bioactive Compounds
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B5670 I-BET 151 hydrochloride1 CitationSummary: BET bromodomain inhibitor -
B5671 JW 67Summary: inhibitor of canonical Wnt pathway signaling -
B5353 DiprenorphineSummary: Non-selective opioid receptor antagonist -
B4571 CH5138303Summary: Hsp90 inhibitor, orally available -
B4755 PI-1840Summary: Chymotrypsin-like (CT-L) inhibitor -
A8896 (+)-MK 801 MaleateSummary: Potent NMDA antagonist -
B4880 WS6Summary: inducer of β cell proliferation -
B5832 Altiratinib1 CitationTarget: FLT3|VEGFR|Trk Receptors|c-MET|Tie-2Summary: c-MET/TIE-2/VEGFR inhibitor -
B5848 KNK437Summary: stress-induced HSP synthesis inhibitor -
B6012 Pexmetinib (ARRY-614)2 CitationTarget: p38|Tie-2Summary: dual inhibitor of p38 MAPK and Tie2/Tek receptor tyrosine kinase

