Bioactive Compounds
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B5910 Rolapitant HClTarget: NK1 ReceptorsSummary: Orally active neurokinin NK1 receptor antagonist. -
B5974 O6-BenzylguanineSummary: Potent MGMT inhibitor -
A8719 ML 239Summary: inhibitor of the breast cancer stem cells -
B5988 TroxerutinSummary: flavonoid -
B6025 DASA-58Summary: activator of pyruvate kinase M2 (PKM2) -
A8723 GSK180Target: Kynurenine-3-monooxygenaseSummary: inhibitor of kynurenine-3-monooxygenase (KMO) -
A8725 UNC3866Summary: a potent antagonist of CBX4 and CBX7 chromodomains -
A3019 AT-406 (SM-406)Summary: IAP inhibitor -
B6044 NCT-501Summary: Aldehyde Dehydrogenase 1A1 (ALDH1A1) inhibitor, Potent and Selective -
B6065 Calcium Ionophore ISummary: Ca2+-selective ionophore

