Bioactive Compounds
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A2942 Masitinib (AB1010)3 CitationTarget: PDGFR|c-Kit|LynSummary: Tyrosine kinase inhibitor, potent and selective -
A2036 Doripenem HydrateTarget: AntibioticSummary: Injectable antibiotic,ultra-broad spectrum -
A1389 WZ4002Summary: Mutant-selective EGFR inhibitor(L858R,T790M), irreversible and potent -
A1980 SNS-032 (BMS-387032)3 CitationTarget: Cyclin-Dependent KinasesSummary: CDK inhibitor -
A1882 Cediranib (AZD217)Target: VEGFRSummary: VEGFR inhibitor receptor,highly potent -
A1736 PA-8242 CitationSummary: Anti-tuberculosis drug -
A1630 Epothilone B (EPO906, Patupilone)Target: Microtubules/TubulinsSummary: Microtubule stabilizing macrolide -
A2487 Odanacatib (MK-0822)Target: CathepsinsSummary: Cathepsin K,potent and selective -
A5932 CandesartanSummary: Angiotensin II receptor 1 (AT1) antagonist -
A5375 TranilastSummary: Angiogenesis inhibitor

