Bioactive Compounds
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A5316 RepaglinideSummary: Kir6 (KATP) channel blocker -
A5343 Ispinesib (SB-715992)Target: KspSummary: Kinesin spindle protein (KSP)inhibitor -
A5919 AZD7762Target: ChkSummary: Checkpoint kinase inhibitor,ATP competitive -
A2033 PQ 4011 CitationSummary: IGF1R inhibitor,potent and cell-permeable -
A2098 PRX-08066 Maleic acidSummary: 5-HT2B receptor antagonist,potent and selective -
A8300 ZCL2781 CitationTarget: Cdc42Summary: Selective Cdc42 inhibitor -
A8303 GNF-5837Target: Trk ReceptorsSummary: Pan-Trk inhibitor -
A8315 NU7441 (KU-57788)4 CitationTarget: PI3K|DNA-PKSummary: DNA-PK inhibitor -
A8320 PF-00562271Target: FAK|Pyk2Summary: FAK/Pyk2 inhibitor,potent and ATP-competitive -
A8329 R42829 CitationSummary: Selective Axl inhibitor

