Bioactive Compounds
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A4317 Apremilast (CC-10004)Target: Phosphodiesterases (PDEs)Summary: PDE4 inhibitor -
A4326 TAK-700 (Orteronel)3 CitationTarget: human lyaseSummary: Human 17,20-lyase inhibitor -
A4342 GimeracilSummary: Dihydropyrimidine dehydrogenase inhibitor -
A1922 Z-VDVAD-FMK3 CitationSummary: Caspase-2 inhibitor -
A3157 AlosetronSummary: 5-HT3 receptor antagonist -
A3266 BS-181Target: Cyclin-Dependent KinasesSummary: CDK7 inhibitor,highly selective -
A3322 Cobimetinib (racemate)Summary: Selective MEK inhibitor -
A3327 CostunolideTarget: FPTase|TelomerasesSummary: Apoptosis inducer -
A3347 Dabrafenib Mesylate (GSK-2118436)Target: RafSummary: Inhibitor of BRAF(V600) mutants -
A3370 Docetaxel TrihydrateSummary: Depolymerisation of microtubules inhibitor

