Bioactive Compounds
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C4880 6,7-dihydroxy BergamottinSummary: potent inhibitor of CYP3A4 -
C4647 β-NicotyrineSummary: cytochrome P450 (CYP) isoforms, CYP2A6 and CYP2A13 inhibitor -
C4837 5(S),6(R)-7-trihydroxymethyl HeptanoateSummary: inhibits leukotriene B4 (LTB4)-induced polymorphonuclear neutrophils (PMN) chemotaxis -
C4756 PF-622Summary: potent, time-dependent, irreversible FAAH inhibitor -
B7875 Adenosine 5-monophosphateSummary: 5'-AMP-activated protein kinase -
C5504 S-methyl-L-Thiocitrulline (hydrochloride)Summary: potent NOS inhibitor -
B5372 HU 308Summary: CB2-receptor agonist -
B5482 MRK 016Summary: GABAA receptor inverse agonist -
B5532 NPS 2390Target: Glutamate (Metabotropic) Group I ReceptorsSummary: group I mGlu antagonist -
B5567 SMER 3Summary: yeast SCF family E3 ubiquitin ligase (SCFMet30) inhibitor
