Bioactive Compounds
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A4060 Geldanamycin2 CitationSummary: Hsp90 inhibitor,potent and specific -
A4154 Olaparib (AZD2281, Ku-0059436)30 CitationSummary: PARP-1/2 inhibitor -
A4112 Barasertib (AZD1152-HQPA)6 CitationTarget: Aurora KinasesSummary: Aurora Kinase B inhibitor, Potent and selective -
A4036 Sitagliptin phosphate monohydrate10 CitationTarget: DPP-4Summary: Potent DPP-4 inhibitor -
A4230 NSC 66811Summary: MDM2 inhibitor -
A4422 L 006235Summary: Cathepsin K inhibitor -
A4412 MDL 281703 CitationTarget: Cathepsins|CalpainsSummary: Calpain and cathepsin B inhibitor, selective -
A4508 ML 228Summary: HIF pathway activator -
A4520 R8-T198wtSummary: Pim-1 kinase inhibitor -
A4538 INCA-6Summary: Selective calcineurin-NFAT signaling inhibitor

