Bioactive Compounds
-
A4170 EPZ004777Target: DOT1LSummary: DOT1L inhibitor -
A4302 Rosiglitazone maleateTarget: Insulin and Insulin-like ReceptorsSummary: PPARγ agonist,high-affinity and selective,potent insulin sensitizer -
A4321 Sildenafil CitrateTarget: Phosphodiesterases (PDEs)Summary: Treat erectile dysfunction and PAH -
A4351 PluriSIn 1 (NSC 14613)Target: Stearoyl-CoA 9-desaturase (SCD-1)Summary: SCD1 inhibitor -
A1924 Z-WEHD-FMK1 CitationSummary: Caspase 5 inhibitor,potent,cell-permeable and irreversible -
A8162 E-64-cTarget: cysteine proteaseSummary: Inhibitor of cysteine proteinases -
A3192 Asenapine hydrochlorideSummary: Atypical antipsychotic -
A3294 CDK9 inhibitor1 CitationTarget: Cyclin-Dependent KinasesSummary: CDK9 inhibitor -
A3384 ElacridarTarget: P-glycoprotein (P-gp)Summary: BCRP inhibitor -
A3583 Matrine1 CitationSummary: Alkaloid found in Sophora plant

