Bioactive Compounds
-
C7197 3-(Methylthio)propionic acid -
A8193 ABT-73735 CitationSummary: BCL-2 protein inhibitor -
A4141 Baricitinib (LY3009104, INCB028050)4 CitationSummary: JAK1/JAK2 inhibitor,selective orally bioavailable -
A4097 CUDC-9072 CitationTarget: Histone Deacetylases (HDACs)|PI3KSummary: Potent PI3K/HDAC inhibitor -
A4100 Droxinostat2 CitationSummary: Selective HDAC inhibitor -
A8206 Darunavir2 CitationSummary: HIV-1 protease inhibitor -
A4124 TAK-901Target: Aurora Kinases|FLT3|Src|JAK|LRRK2|Hck|FGR|YES|Fyn|ARGSummary: Novel Aurora A/B inhibitor -
A4340 PimobendanTarget: Phosphodiesterases (PDEs)Summary: Selective PDE3 inhibitor.Ca2+ channel sensitizer -
A4388 XL-8881 CitationTarget: HSP90Summary: Hsp90 inhibitor -
A1501 Mca-Pro-Leu-NH2Summary: Substrate of matrix metalloproteinases assay
