Bioactive Compounds
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A4077 DabigatranSummary: A potent, reversible direct thrombin inhibitor with core bioactivity of inhibiting thrombus formation. -
A4157 Iniparib (BSI-201)Summary: PARP1 inhibitor,intravenously adminsitered -
A2606 Epoxomicin35 CitationSummary: proteasome inhibitor -
A4038 Alogliptin (SYR-322)1 CitationTarget: DPP-4Summary: DPP-4 inhibitor,potent and highly selective -
A4114 MLN8054Target: Aurora KinasesSummary: Aurora A inhibitor -
A4211 Lenalidomide (CC-5013)Target: angiogenesisSummary: Antineoplastic agent,inhibits angiogenesis -
A4206 Pifithrin-α (PFTα)6 CitationTarget: p53Summary: p53 inhibitor -
A4170 EPZ004777Target: DOT1LSummary: DOT1L inhibitor -
A4302 Rosiglitazone maleateTarget: Insulin and Insulin-like ReceptorsSummary: PPARγ agonist,high-affinity and selective,potent insulin sensitizer -
A4321 Sildenafil CitrateTarget: Phosphodiesterases (PDEs)Summary: Treat erectile dysfunction and PAH

