Bioactive Compounds
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B2184 GDC-0980 (RG7422)Summary: Class I PI3K inhibitor for PI3Kα/β/δ/γ -
B1621 TAK-733Target: MEKSummary: MEK allosteric site inhibitor -
B1303 Amsacrine hydrochlorideSummary: Topoisomerase 2 inhibitor -
C5615 MMP-2 Inhibitor ISummary: reversible inhibitor of matrix metalloproteinase (MMP)-2 -
A1047 Angiotensin 1/2 (1-5)Summary: Vasoconstrictor -
B8540 TBK1/IKKε-IN-5Summary: Dual TBK1 and IKKε inhibitor -
B6128 Fenofibric acidSummary: ppar inhibitor, lipid-lowering agent -
B6188 Pamapimod (R-1503, Ro4402257)Summary: p38 MAPK inhibitor -
B6193 AMG 337Summary: MET inhibitor -
B7804 AG-221 (Enasidenib)1 CitationSummary: mutant isocitrate dehydrogenase 2 (IDH2) inhibitor

