Bioactive Compounds
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A8320 PF-00562271Target: FAK|Pyk2Summary: FAK/Pyk2 inhibitor,potent and ATP-competitive -
A8329 R42829 CitationSummary: Selective Axl inhibitor -
A8444 GW3965 HClSummary: LXR agonist, selective and orally active -
A8519 SB705498Summary: TRPV1 antagonist,potent and selective -
A8542 Triflurdine (Viroptic)Summary: Anti-herpesvirus antiviral drug -
A8402 Conivaptan HClSummary: Vasopressin receptor antagonist -
A8407 Dibucaine (Cinchocaine) HClSummary: Sodium channel inhibitor -
A8610 6,2',4'-TrimethoxyflavoneTarget: Aryl hydrocarbon receptors (AHRs)Summary: Aryl hydrocarbon receptor antagonist -
A8660 Cilengitide5 CitationTarget: IntegrinsSummary: Integrin inhibitor for αvβ3 and αvβ5 -
A8666 TFLLR-NH2Summary: PAR1 selective agonist
