Bioactive Compounds
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B1189 SAR7334Summary: Potent TRPC6 inhibitor -
B1261 Deltarasin hydrochlorideSummary: inhibitor of KRAS-PDEδ interaction, potent and selective -
B1298 K145Target: Sphingosine kinases (SphKs)Summary: SphK2 inhibitor -
B1079 BMS-303141Target: ATP Citrate LyasesSummary: ATP-citrate lyase inhibitor,potent -
B2083 Caspofungin Acetate1 CitationSummary: antifungal lipopeptide compound -
B1931 Dimethyl FumarateSummary: nuclear factor (erythroid-derived)-like 2 (Nrf2) pathway activator -
B1225 Posaconazole hydrateSummary: C14ɑ demethylase inhibitor -
B1463 KPT-276Target: nuclear export|CRM1Summary: inhibitor of nuclear export (SINE) and CRM1, orally bioavailable -
B1180 S1RA hydrochlorideSummary: σ1R antagonist -
B1528 XL335Target: Farnesoid X receptors (FXRs)Summary: FXR agonist

