Bioactive Compounds
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A2597 Brivanib (BMS-540215)Target: VEGFR|FGFR|Flk1Summary: VEGFR-2 inhibitor,ATP-competitive -
A1845 Canertinib (CI-1033)Summary: HER family tyrosine kinase inhibitor -
A5827 AM12412 CitationSummary: Cannabinoid CB2 receptor agonist,potent and selective -
A8308 PH-7978041 CitationSummary: P38 MAP kinase inhibitor, potent and selective -
A8341 Go 6976Target: PKCSummary: PKCα/PKCβ1 inhibitor -
A8436 GabapentinSummary: GABA enhancer -
A8441 GSK4613643 CitationTarget: PLKSummary: Plk1 inhibitor -
A8454 Istradefylline (KW-6002)Target: Adenosine A2A ReceptorsSummary: Selective A2A receptor antagonist -
A8456 JTC-801Target: NOP ReceptorsSummary: KOR-3 (NOP) receptor antagonist -
A8504 Pitavastatin Calcium1 CitationTarget: HMG-CoA ReductasesSummary: Enzyme HMGCR inhibitor

