Bioactive Compounds
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A4049 Marimastat1 CitationTarget: MMPSummary: MMPs inhibitor,board spectrum -
A2586 Nafamostat Mesylate(FUT-175)Summary: Serine protease inhibitor -
A4219 Birinapant (TL32711)9 CitationSummary: Potent XIAP/cIAP1 antagonist -
A1909 BIX 012942 CitationTarget: G9aSummary: G9a and GLP inhibitor -
A1913 RG 1083 CitationTarget: DNA MethyltransferasesSummary: DNA methyltransferase inhibitor -
A4316 KetoconazoleTarget: Cytochrome P450 (CYP450)Summary: Inhibitor of cyclosporine oxidase and testosterone 6 beta-hydroxylase -
A4322 ClarithromycinTarget: Cytochrome P450 (CYP450)Summary: CYP3A inhibitor, potent -
A4333 CPI-6136 CitationTarget: Pyruvate dehydrogenases (PDH)Summary: PDH/α-KGDH inhibitor -
A4335 MildronateTarget: Hydroxylases|carnitine reabsorptionSummary: GBB hydroxylase inhibitor -
A4353 PyrimethamineSummary: DHFR inhibitor

