Transferase
- B5729 GPP 78 hydrochlorideSummary: NAMPT inhibitor
- B5602 GGsTopSummary: γ-glutamyl transpeptidase (GGT) inhibitor, novel and irreversible
- B5521 LY 78335Summary: phenylethanolamine-N-methyltransferase (PNMT) inhibitor
- B5006 OR-486Summary: inhibitor of catechol-O-methyl-transferase
- B3703 LB42708Target: FtaseSummary: Selective FTase inhibitor
- A4384 PF-04620110Summary: DGAT-1 inhibitor,potent and selective
- A4383 TolcaponeTarget: Catechol O-Methyltransferase (COMT)Summary: COMT inhibitor
- A4382 A922500Target: DGATSummary: DGAT-1 inhibitor
- A4381 FK866 (APO866)9 CitationTarget: NamptSummary: NAMPT inhibitor, non-competitive, highly specific
- A4379 LonafarnibTarget: FPTaseSummary: Ftase inhibitor,potent and selective