EGFR
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A3256 BMS-690514Summary: HER/EGFR inhibitor -
A2822 AC480 (BMS-599626)Target: EGFRSummary: HER1/2 inhibitor,selective and efficacious -
A2689 ButeinTarget: Src|STAT|EGFR|Angiotensin-Converting Enzymes (ACEs)|5-Lipoxygenases|PTK|enoyl-acyl-carrier protein reductaseSummary: Protein kinase inhibitor -
A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: HER2 inhibitor,potent and selective -
A2024 PD168393Target: PDGFR|FGFR|EGFR|PKC|insulinSummary: EGFR inhibitor -
A1845 Canertinib (CI-1033)Summary: HER family tyrosine kinase inhibitor -
A1835 Pelitinib (EKB-569)Summary: EGFR inhibitor,potent and irreversible -
A1393 WZ8040Target: EGFRSummary: EGFR T790M inhibitor,irreversible amd potent -
A1389 WZ4002Summary: Mutant-selective EGFR inhibitor(L858R,T790M), irreversible and potent -
A1367 ALK-IN-1Summary: Anaplastic lymphoma kinase (ALK) inhibitor

